Bophelo, Litokisetso
"Simvastatin": ulasan pelanggan, ho bonahala hore li sebelisoe, theko le analogues
Ke hobane'ng ha Ke hloka litlhare "Simvastatin"? Testimonials ka lithethefatsi li tla fanoa e nyenyane ho feta. Re boetse re u bolella mabapi le lithethefatsi ena e fumaneha ka sebōpeho sa eo a nang le matšoao, litla-morao 'me contraindications counterparts, hakaakang ka ho fana, kamoo e lokela ho hantle e sebelisoa le joalo-joalo. D'.
Ambalaji, Product foromo le sebopeho
Lithethefatsi "Simvastatin" tsoela pele Sale mokgwa wa matlapa. Ba na le ho potoloha biconvex sebopeho le letšoao ka lehlakoreng le leng, hammoho le tšoeu. matlapa a tlotsitsoeng, matlapa a joalo na le 10 mg, ea simvastatin. Hape moriana o akarelletsa ho dikarolo ea thusang ka butylhydroxyanisole, lactose, magnesium stearate, starch prozhelatinizirovannogo, talc, le microcrystalline selulose.
Ka sephutheloana ya, o ka reka moriana "Simvastatin"? Bontšang bakeng sa tshebediso ya chelete boletsweng ditaelo, e leng e tse pakete ea lebokoso. Ho boetse ho behoa le machachetsi a mabeli a nkile matlapa (likotoana tse 10).
litla diokobatsi
Joang lithethefatsi "Simvastatin"? litsebi Guest bontša hore lipid-theola lithethefatsi ena. E ya hlahiswa maiketsetso.
Nkoa e le oa moemeli ke kopanele tšebeletsong lactone. Ho batho, e le hydrolyzed, 'me hamorao o ile a bopa e hydroxy-acid e sehlahisoa.
Tšebeliso ea lithethefatsi le ha a bake bokella chefo. Ho ka potlako metabolized le ho akarelletsa'ng dithulaganyo ngata synthesizing.
The thepa ya moriana
Seo thepa ea meriana "Simvastatin"? Reviews bolela hore sesebelisoa sena se ba thusa ho fokotsa maemo lero la mali ea triglycerides, palo yohle k'holeseterole le tlase segokanyipalo lipoprotein.
Phello phekola ka mor'a o qala ho noa lithethefatsi le hlaha ka hare ho ka libeke tse peli. Ketso ea lithethefatsi ea sala e tsitsitseng bakeng sa nako ya kalafo ena. Ka mor'a ho hlakoloa ha matlapa k'holeseterole boemo ba butle-butle o khutlela ho tshebetso ea pele.
Pharmacokinetics
lithethefatsi "Simvastatin" nka nako e kae ba ananelang? litsebi Guest bolela hore absorption ea chelete e phahameng haholo. Holim 'a fumana meriana ka mahloriso lona phahameng ka ho fetisisa ea mali e ile ea fihla ka mor'a lihora tse 1.5-3 le e fokotsehile ka 90% ka mor'a ka 12 lihora tse. Ho buisana le lero la mali le se ka bang 95%.
The metabolism tsa lithethefatsi sebete. Halofo ea bophelo ba metabolites ke lihora tse peli.
Di behilwe moriana o le mantle hammoho le ka ho liphio.
Lithethefatsi "Simvastatin": bontšang bakeng sa tšebeliso
Tsa chelete e kgothaletswa bakeng sa ho sebelisoa hypercholesterolemia, 'me lefu le gogoga pelo. Ho laela moriana joalo lokela ho feela ba ngaka ka mor'a ho hlahloba ka ea tsa bongaka.
Kahoo, ka Leha ho le joalo u ka nka matlapa "Simvastatin"? From hore na ho bolela'ng abetsoe? Ho ea ka litaelo tseo, moriana buelloa ha:
- hypercholesterolemia mathomo;
- le katleho ha lijo le tlaase k'holeseterole lijo le tsereletsi tse ling batho bao e seng lithethefatsi (ho lahleheloa ke boima ba 'mele, ho ikoetlisa) ka bakuli ba atherosclerosis gogoga;
- kopantswe hypertriglyceridemia le hypercholesterolemia, eo e sa a lokisa mejaro 'meleng le ho ja e khethehileng.
Ka seo maemong a mang e beuweng meriana "Simvastatin"? Bontšang bakeng sa tshebediso ya sesebelisoa see hona joale:
- thibelo ea myocardial infarction;
- fokotsa kotsi ea maloetse ea pelo (mohlala, e fetang ischemic tlhaselo kapa leqeba);
- kholofalo ea atherosclerosis ka lijaneng gogoga.
Contraindications
Hona joale hore u tseba seo meriana e hlophisitsweng "Simvastatin". Ho bonahala lebaka la ho sebelisa oa sesebelisoa sa di hlahiswa mona ka hodimo. Leha ho le joalo, lithethefatsi ena ho na le contraindications. Boemo latelang e sebetsa ho bona:
- lefu mesifa (kapa ho thoeng myopathy);
- lefu sebete etsahalang mohato a sebetsang a;
- ba lilemo li 18;
- phehellang bophahamo ba enzyme sebete (ho akarelletsa le etiology tsejoeng);
- hypersensitivity ho lithethefatsi kapa ka ho le metsoako e ka bomong (ho akarelletsa le ho se mamellane lactose);
- hypersensitivity ho ka mekhoa e meng ea statin letoto lena.
Hloko ho lokisetsa baeti ba fihlelang
Moriana o "Simvastatin", theko ea eona e bontšitsoeng tlaase mona, ka hloko ho khetheha e ileng ea fuoa bakuli ba sebelisang joala hampe, hammoho le batho ba latelang lekala transplantation (ka phekolo immunosuppressive).
Ho feta moo, ka taba ena e bolela ka tlhokomelo e entsweng ka maemo a isang ho ntshetsopele ya ho hloleha renal (mohlala, hypotension, mafu a hlobaetsang le a tlhaho a tšoaetsanoang, fokotswa, kapa, ho fapana le hoo, e ile ea eketseha tonus ya dinama tse nyenyane tse mesifa, a bolela hore tshilong ya dijo le endocrine maloetse, lefu la sethoathoa, meferefere electrolyte ho leka-lekana, ho buoa, ho akarelletsa le meno le ho sithabela).
Lithethefatsi "Simvastatin": tšebeliso le litekanyetso li behoa
Nkoa pele ho qapa phekolo bolela mamello o tla feta tekanyetso hypolipidemic lijo. Tshohanyetso, e lokela ho lateloa ho pholletsa le 'nete hore ea phekolo.
"Simvastatin" Letlapa laolwa hang letsatsi le letsatsi ka shoalane. Ha a ntse a ho noa meriana ena lokela ho tsamaisane le tshebediso ya ea lijo.
The kgothaletswa litekanyetso li behoa bakeng sa kalafo lithethefatsi tsa hypercholesterolemia ke 10-80 mg, ka ho ya ka letsatsi.
liphetoho lethal dose lokela ho ho phethahatsoa ka dikgao tsa khoeli le khoeli. Ntlha ea pele, le mamello lokela ho nka 10 mg,, moo 20, 30 'me joalo-joalo. D. Maemong a mangata ho homolog phekolo e le hantle e fumana ha fumana 20 mg, ea moriana.
The litekanyetso li behoa ea ea lithethefatsi e ho itšetlehile ka lilemo tsa mokuli a se, boemo ba lona le tse ling tse joalo. Tabeng ena, joalo pheko lokela ho thonya ngaka, ka mor'a ho hlahloba mokuli le ho hlahloba ka ea meriana.
liphetoho tse bohloko
Joalokaha eka ke ka leha e le efe ea lithethefatsi, moriana o "simvastatin" o boetse o na le liphello. Har'a atileng ka ho fetisisa ke e latelang:
- Mpeng bohloko, lefu la sebete, pipitlelano, pancreatitis, flatulence, ho hlatsa, phahameng sebete enzyme, letšollo, le ho nyekeloa ke pelo.
- Asthenic lefu, phytoteratology kutloisiso ea tatso, hlooho e opang, pono thothofatsang, molikoalikoane, ho neuropathy pheriferale, lefu la ho hlobaela, paresthesia, cramps mesifa.
- Angioedema, eosinophilia, polymyalgia rheumatica, urticaria, lupus-joaloka lefu, vasculitis, dyspnea, thrombocytopenia, mahlaseli a chesang, e ile ea eketseha erythrocyte sedimentation sekhahla, Flushing tsa letlalo, feberu, photosensitivity, ramatiki.
- Letlalo lekhopho, alopecia, dermatomyositis, ho hlohlona.
- cramps Myopathy, rhabdomyolysis, myalgia, bofokoli, mesifa.
- Khaello ea mali, fokotswa potency, pelo, renal ho hloleha (a hlobaetsang le).
litaelo khethehileng bakeng sa kamohelo moriana o
Pele o sebedisa sehlahiswa o lokela ho bala litaelo ka hloko. E bolela hore:
- pele qala ha phekolo e ho hlokahala hore ho khanna thuto ea sebete;
- lithethefatsi "Simvastatin" ha aa lokela ho ho nkoa ka ka taba ea ho hloleha renal le e kotsi ea ho rhabdomyolysis a ekeletsoa;
- meriana e ka ba le liphello tse bohloko ka lesea la;
- ho e sa kgothaletswa ho nka lipilisi ho basali ba ho ba le bana lilemo ba sa sebelise lithibela-pelehi;
- nakong kalafo ha lia lokela ho sebelisoa hampe le joala bo bongata;
- nakong phekolo, mokuli lokela ho iphaphatha le seratsoana hypolipidemic;
- tsoa hong baeti ba fihlelang ho ya lero grapefruit ka khona ho ntlafatsa tekanyo ea ho tiea a itšoare lehlakoreng;
- ho lokisetsa le ka ho ba e atlehang e le monotherapy, 'me hammoho le ho sebelisa ha sequestrants bile acid e.
Analogs le theko ea lithethefatsi e
Hona joale u tseba hore ke lithethefatsi "Simvastatin". Analogues, theko ea phekolo ena o tla fuoa ho hona joale.
Haeba ho ke ke kopo khonehe ea mokhoa ona ka nkeloa sebaka ke lithethefatsi tse ling tse kang "Simvakard", "Avestatin", "Holvasim", "Aktalipid", "Sinkard", "Aterostat", "Simplakor", "Vasilip", "Simli" "Vero -Simvastatin "," Simgal "," Zovatin "," Simvor "," Zocor "," Simvastol "," Zorstat "," Simvalimit "," Ovenkor "," Simvakol "," Simvageksal "le sa t. d '.
lithethefatsi theko "Simvastatin" ha se phahameng haholo 'me ke ka 240 li-ruble bakeng matlapa 20.
Reviews of moriana o
bakuli ba bangata ba kile "Simvastatin" matlapa a, hlokomela bokgoni lona phahameng. Lithethefatsi ke ka potlako lowers k'holeseterole, ho thibela ntshetsopele ya mafu a sa tšoaneng.
Leha ho le joalo, ba bang ba ba teng bakuling ba sa thabang eo ho fetile mora kalafo k'holeseterole boemo ba hlaha hape 'me hangata tabeng ea ho ya motheo wa.
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