Bophelo, Litokisetso
"Antabuse" lipilisi. Reviews, theko motataisi
E bitsoa ho lemalla joala ke lefu le e tšoauoa ka ho lemalla ho ethanol le ho itšetleha 'meleng le kelellong ho eona. Ea mofuta ona e le ho hlekefetsa. Ka puso ena, ho lahleheloa ke matla a ho laola chelete joala tahiloe eketsa mamello ho e (ho fihlela ka khotsofalo e joala kamehla eketseha lethal dose) le a khaotsa ho tsuba lefu le hlaha, ho ama litho tse ka hare le hlaha ea thisa hlooho.
Bakuli ba nang le bokhoba ba tahi, e bitsoang makhoba a tahi. Tšoara le lefu lena e lokela ho ba kelellong le 'meleng. hangata haholo, lingaka ho laela lithethefatsi eo ho batho "Antabuse". Litaelo tsa tšebeliso, theko ea meriana, ulasan pelanggan tsa bongaka di bontšitsoeng tlaase mona.
Paka, sebopeho, le tlhaloso ea sebopeho
Ka seo theha lithethefatsi e rekiswa "Antabuse"? Testimonials tlaleha hore joalo pheko ka rekoa ka mokgwa wa e tšoeu, potoloha matlapa effervescent. Ba bataletseng, beveled bohale, kotsi le tšoauoa «CD» le «C» ka mahlakoreng a fapaneng le likotsi.
Sebopeho sa meriana ena e kenyeletsa disulfiram. Ntle ho, ho lokisetsa ho na le poone starch, povidone, sodium hydrogencarbonate, acid e tartaric, colloidal silicon e dioxide, talc, microcrystalline selulose le magnesium stearate.
Tablets "Antabuse" kenngoa ka lik'hontheinara polasetiki le ka gare ga mapokisana lebokoso.
litšobotsi tse pharmacodynamic
ke lithethefatsi "Antabuse" ke efe? e re Manual hore sena se bolela antialcoholic. Ho thibela acetaldehyde dehydrogenase, e amehang ka metabolism ea ethanol. Lieha thulaganyou e lona ho kena moea o etsa hore ho bokella joala le ntshetsopele ya botahoa matla, lateloa ke maikutlo a boima ka bohloko throbbing le lerata ka hlooho, tachycardia, palpitation, ho fokotseha ha khatello ea mali, ho nyekoa ke pelo, pono thothofatsang le ho hlatsa.
Ho latela litsebi, matšoao ana a sa thabiseng kenya letsoho hore ho ho hōla ha masusu reflex hloile ho noa joala.
thepa pharmacokinetic
Joang absorption ea "Antabuse" lithethefatsi? Manual e bontša hore lithethefatsi e ananelang 70-80%. O haholo qhibilihang ka har'a ka lipids le atisa ho ipokellela ka depo mafura.
Ntho mafolofolo le moemeli ka potlako haholo metabolized, ea fella ka hore metabolite fetohe - methylene Ester dietiltiokarbaminovoy acid e. Lona concentrations tlhōrō mali ikemiselitse mora 4 H. Le hoja mosebetsi mabapi le acetaldehyde dehydrogenase e ketekoa feela ka mor'a matsatsi a mararo.
The halofo ea bophelo ea lithethefatsi ke lihora tse 10. Ho feta moo, mosebetsi lona khahlanong aldehyde dehydrogenase phehella nako e telele haholo. Ka lebaka leo, ka mor'a hore hlakoloa ha phello ea matlapa ao ba a hlokomela ka ho eketsehileng matsatsi a 7-14.
Lithethefatsi hlaha ka moroto, 'me karolo e' ngoe ka mala le moea exhaled.
ya litatoli na
Maemong a mang, le lithethefatsi atlehang ka ho fetisisa itshwara "Antabuse"? Reviews ba tlalehile hore setsing sena ho pharaletseng sebediswa bakeng sa thibelo ea khutlela mokhoeng ea ho phekola ba itšetleha joala le ho lemalla joala.
Contraindications
Ha ua lokela ho nka "Antabuse" Letlapa? Guest litsebi re nahana ka lithethefatsi ha baa lokela ho e beuweng haeba:
- glaucoma;
- neuritis tsa optic le methapo ea kutlo utluwang;
- lefuba methapo;
- pelo le vascular mafu (mohlala, poso-infarction bolela, a bontša cardiosclerosis, atherosclerosis likepe bokong, hypertension lefu, aortic aneurysm);
- polyneuritis se hlahang ho yona efe kapa efe;
- lefu la tsoekere;
- emphysema, bronchial asma;
- thyrotoxicosis;
- lefu la kelello, lefu la sethoathoa 'me lefu epileptiform;
- hlahala;
- e amanang le sebete haholo 'me ho hloleha renal;
- mafu a hematopoiesis;
- exacerbation ea boloetse peptic seso;
- bokhachane;
- hypersensitivity.
Hape ela hloko hore lithethefatsi ena ke contraindications a lekanyelitsoeng:
- ba lilemo li 60;
- liphello tsa ho se leqeba le matšoao a barrel;
- peptic seso (ho akarelletsa le ho bolelang ho leballa motho);
- precipitates e psychosis.
Lithethefatsi "Antabuse": litaelo tsa tšebeliso
-Ba khahlanong le ho noa joala pilisi theko thathamisitsoeng qetellong ea sehlooho se reng. Lokela ho nka bona ka hare ½ pele qhalwa ho ya ka khalase ea metsi.
Ka tloaelo, lingaka ho laela 200-500 mg, ea lithethefatsi hang kapa habeli ka letsatsi. Ka mor'a matsatsi a 7, le be le bonnete ba hore ho qeta teko disulfiram-joala. Ka e tšoanang le baeti ba fihlelang ho ba 500 mg, ea dino moriana o le mamello 20-30 di ml ea vodka. Ha ba itšoara joang ke fokola, joale eketsa lethal dose ea joala ho 20 di ml.
teko ena e phetoa ka makhetlo a mangata. Hamorao ballroom balletsweng tokiso litekanyetso li behoa ea 200 mg, letsatsi le letsatsi bakeng sa ho lilemo tse 1-3.
liphetoho tse bohloko
Tablets "Antabuse", eo dikatlholo di hlahiswa mona ka tlase ho ka etsa hore liphello tse latelang lehlakoreng:
- lefu la sebete, asthenia, tšepe tatso ka molomo;
- cutaneous liponahatso, maoto polyneuritis;
- ho lahleheloa, boko ho ruruha, ho tšoaroa ke hlooho;
- myocardial infarction, cardiac arrhythmias;
- ho hema ho hloleha, pelo le methapo putlama;
- optic neuritis, bokong lijana thrombosis;
- psychoses, angina.
Moriana o "Antabuse": ulasan pelanggan tsa lingaka le theko
Litsenyehelo tsa ho ba matlapa-ba khahlanong le ho noa joala e ka 450-600 li-ruble (ho itšetlehile ka lethal dose 'me chelete ka pakete).
Lingaka li ba ho hlalosa lithethefatsi tse joalo, hang-hang o ile a lemosa la mathata a tebileng tsa hore ka etsahala ka mamello ka morao ho tla nka. Ka lebaka leo, ka tieo thibetsoe ho tšoara kapa ua e le lekunutu ho tloha ba le mamello.
Ho lokela ho hlokomeloe hore litsebi tse ngata lia lumela hore lithethefatsi e atlehang eo hatella ea ho lakatsa ho noa lino tse tahang, ha ho na. Le mokhoa ona ha phekolo. E mpa feela e khothalletsa e kokobetse tsitsitseng.
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