BopheloLitokisetso

"Estrozhel": litaelo bakeng sa ho sebelisoa, tlhaloso ya ba lokisetsa ho, analogs, litla-morao

Ho na sephiri le bakeng sa lefu climacteric tšoauoa ka autonomic-vascular, kelellong le tshilong ya dijo le endocrine mafu a hlahang ke motho oa bong fairer ka kakaretso lilemo involution ea phelang, hammoho le ka semelo sa pheliso butle-butle mosebetsi hormonal popelo.

Ka nako ena e thata bakeng sa basali ba kamehla ba ikutloe flushes chesang ho hlooho, 'mele oa ka holimo le matsoho.

Ho phaella moo, matšoao a menopause kenyeletsa teneha ka tsela e feteletseng, lefu la ho hlobaela, ho tepella maikutlo, ho fokola le boikutlo tšabo e sa khaotseng. Hangata, batho ba bong bo fairer fetola takatso ea botona kapa sitisa migraine, molikoalikoane, hammoho le ho ba le tsela e feteletseng ho fufuleloa, edema le vasospasm.

Ho fokotsa boemo ba mosali eo, lik'hamphani lithethefatsi ba ile ba qala ho hlahisa lithethefatsi protivoklimaktericheskie. The atlehang ka ho fetisisa ea bana ba kenyeletsa moriana kang "Estrozhel". Reviews (nakong menopause ke mokhoa balletsweng hangata haholo) basebelisi tla tšohloa mona ka tlase. U tla boela u ithute ho sebelisa lithethefatsi o ile a re, hakaakang ka ho fana, 'me joalo-joalo.

Tlhaloso, sebopeho, ambalaji le mofuta o sa lokolloe

rekiswa moriana "Estrozhel" Ka mofuta o eng? Reviews of basali bolela hore sethethefatsi ka fumanoa ka mokgwa wa e transdermal gel. Ho colorless, pepeneneng, mme o na le monko oa ethanol.

The a sebetsang a motsoako oa moemeli ena nka khato estradiol. E le metsoako ea thusang moriana o na le carbomer, ethanol, trolamine le metsi a hloekisitsoeng.

Ho lokisetsa "Estrozhel" (gel) e rekiswa ka methapo ea aluminium. Hape e ne e akarelletsa ke applicator khethehileng ho aba.

makgetheng diokobatsi

ke gel "Estrozhel" ke efe? Litaelo ka kōpo ea ho bontša hore ke moemeli hormonal, e leng se etsang bakeng sa ho haella ha estrogen bananeng 'meleng oa mosali.

Thanks ho entsoe a sebetsang a moriana ona o mosebetsi estrogenic. E reretsoe feela bakeng sa kopo Link kapa lihlooho tsa puisano.

Ka ho phekola setsing sena bong fairer haholo fokotswa matšoao a lefu menopausal, ho akarelletsa le ho tepella maikutlo, lekhopho, flushes chesang le omile bosaling.

Ka bokgoni lona ea tleleniki ea ho phekola matšoao postmenopausal nkoa meriana ha e le fe ho kalafo le estrogen bananeng phekolo molomo. Ho feta moo, ha u sebelisa sesebelisoa sena bakuli menopausal tšoauoa slowing tsa dithulaganyo hore fokotsa segokanyipalo sa ea dinama tse nyenyane tse masapo.

Hape o ile a qeta phekolo thusa fokotsa palo yohle k'holeseterole.

Re ke ke ra bolela hore lithethefatsi "Estrozhel", theko ea eona e bontšitsoeng tlaase mona, o na procoagulant bokgoni. Ho fokotsa palo ea antithrombin III le eketsa e amanang le sebete tswakana ba mahlahana K-itšetlehileng ka mali hoama.

thepa pharmacokinetic

Hore na meriana e ananelang "Estrozhel"? Reviews litsebi re ka mor'a ho sebelisa gel e etsahalang ka potlako haholo evaporating ethanol e, oo ka oona estradiol hang-hang le kenella ka hare ho letlalo. A karolo e khōlō ea lithethefatsi ho hang-hang kena ajoa systemic, 'me e nyenyane - e bolokoa ka mafura subcutaneous, eo hape a lokolloa butle.

Ka mor'a ho sebelisa ea moo ba gel palo e kahodimodimo ea mahloriso ea estradiol ka mali ba ile ba hlokomela ka mor'a metsotso e 180-240. The bioavailability ea lithethefatsi ke 82%.

O ne a nka moriana o ha e tlas'a phello ea "fetisetsana pele", eo e fana ka a godimo a lero la mali mahloriso tsa estradiol ha ho bapisoa le analogues molomo.

A khaotsa ho tsuba ba estradiol le phetoho lona tshilong ya dijo ka ho tšoana le tseo ho tšoanang estrogen bananeng tlhaho.

Bontšang bakeng sa kopo ya ba lokisetsa ho Link

Bakeng sa hore na morero oa lithethefatsi "Estrozhel" ka sebelisoa? Litaelo bakeng sa ho sebelisoa li bontša hore pheko ena e kgothaletswa ho fokotsa kapa ho felisa matšoao a ho lefu climacteric, ho akarelletsa le artificially hlohlelletsoa menopause. Ho phaella moo, lithethefatsi potso e atisa ho sebediswa bakeng sa ho thibela le kalafo ea osteoporosis nakong menopause.

Contraindications

Na u se u tseba hore ha ua lokela ho sebelisa gel "Estrozhel"? Litaelo bakeng sa ho sebelisoa e tlaleha hore ho contraindications ho feletseng oa sesebelisoa se akarelletsa maemo a kang a latelang:

  • Male rotor lefu;
  • ischemic kapa haemorrhagic leqeba;
  • hlobaetsang thrombophlebitis kapa thromboembolism;
  • nakong ea bokhachane;
  • mali uterine se hlahang ho yona undetermined;
  • renal ho hloleha;
  • kanyeso;

  • ; Johnson - lefu Dubin
  • estrogen bananeng-itšetlehileng ka malignancies kapa belaelloa ka hore boteng ba bona;
  • hypersensitivity;
  • nang kotsi kapa bolaeang lihlahala tsa pituitary ea;
  • Nka Lintho ka Botebo lefu sebete ka mohato hlobaetsang, lihlahala sebete, 'me nyooko.

Hloko tshebediso ya moriana o le

Ha ke lokela ho sebelisa gel "Estrozhel" hlokolosi feteletseng? Guest litsebi re'ng ka maemo a latelang:

  • leiomyoma;
  • gogoga mothapo lefu;
  • endometriosis;
  • meferefere ea mosebetsi sebete;
  • pancreatitis;
  • lefu la tsoekere;
  • migraine;
  • sethoathoa;
  • asma;
  • lelapa hyperlipoproteinemia;
  • e amanang le sebete porphyria;
  • hlabang lefu ea tsamaiso ea ho ikatisa ka ho kopanela liphate fairer;
  • o ile a re pele nyooko, ho akarelletsa le ponahalo ea eona e leng tsela ea ho ima ho qetela;
  • trombozay, thrombophlebitis kapa thromboembolism (bapisoa estrogen bananeng kalafo);
  • kgatelelo ya madi ka matla;
  • bolwetse gallbladder le cholelithiasis (histori);
  • hypercalcemia amanang le metastases lesapo la letsoele dinama tse nyenyane tse ka lihlahala;
  • mafu a ho potoloha ha mali.

Gel "Estrozhel": litaelo tsa tšebeliso

Ba ne ba nka ho lokisetsa e sebediswa ka lihlooho feela. Tabeng ena e sebelisoa tswelela pele kapa cyclically. Nako ea phekolo le litekanyetso li behoa ea ea lithethefatsi a khetha le batho ka bomong.

lethal dose e mong oa gel "Estrozhel" (2,5 g) e na le 1.5 mg, ea estradiol.

Ea ho phekola matšoao menopause bontša lahloang ho sebelisa lithethefatsi ka letsatsi ka palo ka lethal dose. The gel ile thinly hasana ho fetela ho letlalo sebakeng sa lumbar sebakeng, forearm, mpa kapa ka mahetla, 'me ba letetse fire lona ka ho feletseng.

sebaka sa letlalo moo moriana o ne a etsa kōpo, ke ke ba le ka tlaase ho e sebakeng oa matsoho bobeli ba mokuli.

Bakeng sa tshebetso e nepahetseng ea dikopo le lebaka atlehang ka ho fetisisa e tsejoang ka ho absorption ea moriana ka mor'a metsotso e 3. Ka nako e tšoanang sa ho pholosa stickiness mora kopo ya lethal dose e le 'ngoe ea lithethefatsi bakeng sa metsotso e 5 bontša ho hloka sebaka sebelisoa ke letlalo.

Sebetsa meriana lokela mokuli (hoseng kapa mantsiboea). Sebelisa gel ke ho hotle ho likoahelo pele clean.

litla-morao

ke eng liphello batleheng etsahala ka mor'a ho sebelisoa ha "Estrozhel" gel? Reviews of basali tlaleha liphello:

  • letlalo ho teneha, letlalo e phallang, ho tšoaroa ke hlooho le migraines;
  • feto-fetoha, 'me ho tsekela;
  • nahanela le ho eketseha ha boholo ba litsoelesa le mammary, bohloko ba bona, menorrhagia, amenorrhea, katleho e kholo tsoa mali;
  • lihlahala ka litsoelesa le mammary, e ile ea eketseha libido, smearing tjhajoloha bosaling, ho akarelletsa le nako intermenstrual;
  • indigestion, nyooko senya obstruction, ho nyekoa ke pelo, ho hlatsa, lefu la sebete, epigastric bohloko, ho ipolaisa tlala, pancreatitis;
  • cholelithiasis, cholestatic nyooko, letšollo, mala cramps, bloating;
  • thromboembolism ikopanye lense se mamellane, liphetoho tse boima ba 'mele, edema pheriferale;
  • eketseha khatello ea mali, kulisa (ho akarelletsa le urticaria le ho hlohlona la letlalo), ikopanye le dermatitis.

Kaofela ha liphello tsena lehlakoreng di bolela hore ena length of. Hangata ba teng ka mekhahlelo ea pele ea phekolo le hoo e ka bang mohla hloka discontinuation ya meriana.

matšoao a overdose

Ho tla etsahala'ng ha e kholo chelete ea lithethefatsi "Estrozhel" (kamoo u ka sebelisang sesebelisoa sena, re ile a re ho ka holimo)? Tabeng ea tekanyetso e phahameng ea moriana o ka nyekeloa ke pelo le mamello le ho hlatsa, hammoho le hlahisa mali uterine. Ka sebopeho sa matšoao a tsena sebelisa gel hang-hang khaotsa.

Sebelisana le lithethefatsi tse ling

Na hoa khoneha ho kopana le lithethefatsi tse ling tse lithethefatsi "Estrozhel" (gel)?

  • Ka kopo e tšoanang le ea mahlahana antihypertensive le hypoglycemic, le anticoagulants ka 'na fokotsa katleho ea bona, e leng hloka hore a review le tsa puso ea dosing.
  • Ha e kopana le "Estrozhelya" le lithethefatsi lipid-theola isang ama haholoanyane tsela eo e qetellang.
  • Ka tšebeliso tsoa hong le lithethefatsi tse inducers tsa microsomal sebete enzyme (mohlala, "rifamycins", "Carbamazepine", "griseofulvin" le barbiturates), lero la mali estradiol a ka fokotseha.
  • Tshebediso ya gel le ho fokotsa ho atleha ha diuretics le li-hormone ho kopanela liphate e motona.
  • Tshebediso tsoa hong ea lithethefatsi, analgesics opioid le lithethefatsi sebediswa bakeng sa thethebatso kakaretso, eketsa metabolism tsa estradiol.
  • Ha e kopana le lithibela-mafu tse itseng (ho akarelletsa le "Rifampicin" le "ampicillin"), hammoho le "phenylbutazone" fokotsa concentrations lero la mali ea estradiol.
  • Tsoa hong kalafo le folic acid le thyroid li-hormone eketsa estradiol litla ho bolela.

likhothaletso itseng

Lithethefatsi "Estrozhel" tšebeliso e tieo thibetsoe nakong ea bokhachane. Ho lokela ho hlokomeloe hore pele kopo ya gel basali e lokela ho ba bonnete ba hore fumana e feletseng gynecological hlahloba. Ka nako e telele ya moriana, ditsamaiso joalo ba lokela ho ho phethahatsoa bonyane hang ka selemo.

Ho ea ka ka dikgothaletso kalafo setsebi se advantageously etsoa hammoho le estradiol, phekolo progestin. Joalo motswako e tla sireletsa endometrium.

Ho lokela ho sireletsa mucosa ea bosading le hara botshehadi, hammoho le letlalo ka letsoele ho tloha ho ka ba nkoa lithethefatsi.

sebelisoa ka nako e telele ea lithethefatsi, ho akarelletsa le tekanyetso e phahameng, ho eketsa kotsi ea letsoele le kankere endometrial.

Ha o batla ho elective buuoa, ea estrogen bananeng phekolo lokela ho khaotsa ho qeta libeke 4-6 pele.

"Estrozhel" ha ea lokela ho sebelisoa nakong ea thero ea bokhachane. Ho lokela ho hlokomeloe hore ho moriana o le mafolo-folo ha dithibela thepa le ha e thibele kemolo.

Lithethefatsi "Estrozhel" le "Utrozhestan" - motswako phethahetse. Ka lebaka la tokisetso ena le boleng ba bophelo ba mokuli nakong menopause haholo ba ntlafala.

litokisetso theko le tšoanang

Ke bokae ka gel "Estrozhel"? Theko ea moemeli ena ke tse ka bang 700 li-ruble. Haeba hlokahala, e ka nkeloa sebaka ke lithethefatsi tse ling tse kang "Estrokad", "Esterlan", "Estrovagin", "Ovestin", "Sinestrol", "Kolpotrofin", "ethinylestradiol", "Elvagin", "Ovipol Clio", "Pauzogest "," Klim "le ba bang.

Reviews basali

Batho ba bong bo fairer ho sebelisa mekhoa ea ho ea liphallelo matšoao menopausal, a mo siea a poeletsotlaleho feela e nepahetseng. Ba ela hloko bokgoni lona phahameng le maqhubu a tse nyenyane le ho tiea tsa litla-morao bapisoa le counterparts molomo.

litšobotsi tse ling tse ntle tsa moriana kenyeletsa loketseng dosing mochine lona, lebaka la ho hloka tackiness mora Tsamaiso le absorption ka potlako ka letlalo.

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