BopheloLitokisetso

Aromatase inhibitors: recensioni, litheko. inhibitors Aromatase ka bodybuilding

Aromatase inhibitors, kapa blockers, - ea mofuta ofe lisebelisoa tse sebelisoang ho fokotsa mahloriso tsa estrogen bananeng, ka mali le eketsa boemo ba folisa gonadotropins le testosterone. dintho tsena di a boela a sebelisa bakeng sa kalafo le thibelo ea gynecomastia motona.

inhibitors Aromatase ka bodybuilding ba atisa ho sebelisoa nakong ea tsela ea steroid anabolic ho:

  • ho ntlafatsa tshebetso ya anabolic hormone maling;
  • thibelo gynecomastia;
  • thibela kgatelelo ya madi;
  • eketsa bump (by felisa phello e mpe ea estrogens);
  • fokotsa estrogen bananeng felisoeng ha a selekane otlwa makwalateng-pituitary-hypothalamus, e isang ho tsosolosa e potlakang.

Ho haha tsela e, o lokela ho Itekanyeng le e le hantle hore tatso ha e ikamahantse le anabolic steroid tsohle. Sebelisa e le lebaka le utloahalang ha tšebeliso ea lihlahisoa tse kang methandrostenolone, methyltestosterone, testosterone le derivatives lona. Hanyenyane tatso Halotestin, boldenone.

katleho

Ka ho fetisisa ba rata le ho fumaneha inhibitors aromatase (bakeng sa behang litholoana hoo e batlang e tšoanang):

sehlooho se reng

(Global sehlooho)

Cha (rekiswang ke bapharmasi)

theko e lekantsoeng

Foromo ya ho lokolloa

Prophylactic bodybuilding

Ha gynecomastia

"Exemestane"

"AROMASIN"

1600 li-ruble.

30 tab ya. 25 mg,

2,5 mg, (matlapa halofo) letsatsi le letsatsi tse ling

25 mg, letsatsi le letsatsi ho fihlela le matšoao liquidation. Ebe litekanyetso li behoa phokotso ho prophylactic.

'Letrozole'

"Letromara" (Farmak).

"Letroza"

"Estrolet"

3200 li-ruble.

1000 li-ruble.

30 tab ya. 2,5 mg,

0.5 mg, (matlapa 1/5) letsatsi le letsatsi tse ling

2,5 mg, letsatsi le letsatsi ho fihlela le matšoao a ho felisoa. Ebe litekanyetso li behoa phokotso ho e thibelang e ka.

"Anastrozole"

"Motse"

"Egistrazol"

"Anastrozole kabhi"

1500 li-ruble.

350 li-ruble.

1300 itlotsa.

28 tab ya. 1 mg,

0.5 mg, (matlapa halofo) letsatsi le letsatsi tse ling

1 mg, letsatsi le letsatsi ho fihlela le matšoao liquidation. phokotso ka ho eketsehileng le litekanyetso li behoa prophylactic.

Re lokela ho hlokomela hore le leka-lekaneng tsa mahloriso tsa estrogen bananeng, na le thuso bakeng sa khōlo e mesifa, leha ho le joalo thibela dosages ho bontšitsoe lintho tse ngata tse amang ho pholosa physiologically hlokahalang boemong ba estrogens motona.

Sebelisa thupelo

Boholo ba baatlelete malapeng sebelisa inhibitors aromatase, sebelisa maqiti a latelang: lithethefatsi li sebelisoa feela ha matšoao pele la gynecomastia (ho hlohlona la nipples e, ho ruruha, redness). Ka bomalimabe, mokhoa ona o ke ke bitsoa homolog.

The tharollo fetisisa kwalwang e nkoa e lekoa estradiol ka bang leshome matsatsi a, ho sebelisa anabolic steroid ka e khutsoanyane halofo bophelo ( "Methandrostenolone", "Testosterone propionate") kapa libeke tse tharo kapa tse 'nè tsa kopo ya o molelele o Ester ( "Sustanon", "Enanthate," "cypionate"). Ho ekelletsa moo balletsweng karolo karolelano "Anastrozole" - 0.5 mg, mong le e mong tse ling tse letsatsi. Ka mor'a matsatsi a leshome, e neng e tšoaretsoe ka and analysis laola ya estradiol le litekanyetso li behoa e fetola ho latela liphello.

Sekisetsa ha ke ho sebelisa tlase le e leka-lekaneng servings "Anastrozole" tsepame maikutlo botho. Haeba mora jwalo kalafo e ba tepeletseng maikutlo, ho hloka taolo ya erectile mosebetsi, libido lerotholi, nako eo o lokela ho fokotsa lethal dose ya.

ho etsa lipatlisiso

Ho hlaha ha e setjhaba cha "letrazole" tlisa sehlahisoa sena ka pele. Ho na le mefuta e fapaneng ya liteko ho paka ho atleha phahameng oa sesebelisoa sena e leng banna. Ho qaloa ho dintho tsamaea le ho phahama ha ho tshwailwe tsa gonadotropin (LH). Behang litekanyetso li behoa e simoloha ho tloha 0,02 mg, (ho phekola ka tlase ka makhetlo a 100): ho ka etsahala ka tsela ea boraro ka tlaase estrogen bananeng mahloriso. 50% "letrozole" felisoa ho 'mele nakong ea matsatsi a 2-4, e le hore a noe le letsatsi. The drawback mantlha e nkoa e le matla a ho maemo e ka tlaase ea estrogen bananeng, esita le ka tekanyetso e nyenyane.

"Anastrozole" ratoang bodybuilding, ka tsela e hlollang ea hae a ithuta ka banna e le mokhoa oa ho fokotsa estradiol. Empirically e ile bontšitse hore ka lethal dose ea 1-0.5 mg, estradiol boemo ba ka 'na fokotseha ka hoo e ka bang 50%. Dealers sehlahisoa sena se ka rekoa ho fihlela ho ka makhetlo a leshome theko e tlaase ho feta famasi ena. Ka megacities kopana theko "Anastrozole kabhi."

Bukeng ea hae, Dr. Mauro G. De Pascal o ile a ngola: "Ho nahana hore estrogens tse thehoa ka lebaka la aromatization ea testosterone kapa tse ling tse anabolic steroid ka mafapha a tsa hypothalamus le boko, ho fokotsa secretion ea luteinizing hormone, 'me, ka lebaka leo, ho hlahisa testosterone." Gilman le Goodman tsebisoa hore poeletsotlaleho e butswe ho ena le bokella tsa estrogen bananeng, ho ena le testosterone. Ka tsela ena, e ile a hlalosa hore inhibitors aromatase ka fokotsa phello inhibitory tsa anabolic mahlahana a ho abelwang karolo ya li-hormone ho kopanela liphate ea botho.

litla-morao

The inhibitors aromatase ke kotsi bakeng sa banna? Rea tseba hore estrogen bananeng ka tekanyetso tlaase na le phello e ntle ka 'mele e motona. Estrogen bananeng hormone eketsa le nkang le bokgoni le ba nahanela ba receptors androgen. Ho feta moo, bona ka bobona ba ba le phello e sireletsang le anabolic.

E bolelang mesifa estrogen bananeng receptor ho feletseng o ile a hlalosa ka Anna Wiik ka ho qaqileng. Ha e le hantle hlile tsotehang blocker lethal dose ka 'na sa hlokahale fokotsa boemo ba estrogen bananeng, e thusa hore ho ho hlaha ha litla-morao tse kang:

  • thibelo ea khōlo ea mesifa;
  • bohloko e kopanetsoeng (arthralgia);
  • bophelo ho senyeha le ho fokotseha ha libido;
  • ho tepella maikutlong;
  • boloetse mali lipid profil (k'holeseterole keketseho e);
  • fokotseha ka matla a masapo.

Subjectively, lithethefatsi le ba molemo ho sa mamelloe batho ho feta "Tamoxifen".

inhibitors tsa tlhaho

Ke tse latelang:

  • caffeine;
  • resveratrol;
  • zinki;
  • bokoali;
  • apigenin;
  • catechins;
  • eriodiktiol.

Ho sebelisoa ha "Anastrozole"

More feta inhibitors e ntle aromatase? lithethefatsi tsena li ka ba hohle sebelisoa ka bodybuilding. Mohlala, "Anastrozole" hlokehang bakeng tshegetsa le go tlotla metsi ka 'mele oa motho le ho thibela ketsahalo ea gynecomastia (hangata e le ka hammoho le oa androgens testosterone le Dianabol mofuta kapa hammoho le finasteride). Empa tabeng ena, le moatlelete fumana hammoho le rarahaneng ee e hlollang ea lithethefatsi e hanetsoeng ho tloha "lethathamo la dintho tse thibetsoeng le mekhoa", ntle le mefuta e fapaneng ea eona ea litla mahareng.

Tshebediso sa laoleheng ea "Anastrozole" baatlelete, jara ka, ka ho khetheha, bodybuilding ka etsa hore arthralgia, asthenia, kapa ho fokotsa le tsamaiso manonyello, hlooho e opang, somnolence. Ke 'nete hore ka linako tse ling a ka hlaha mathata thromboembolic le ho ntshetsa pele lichapo.

Ka "Anastrozole" Boholo e se e ngotsweng ka lingoliloeng tsa baatlelete ka lithethefatsi kotsi haholo. Empa litla hōle le hang-hang ka baeti ba fihlelang ho sona e ka ba tsejoa esale pele haholo le tse bohloko. Ka sebele, haeba feela ho nka letlapa le leng (1 mg,) letsatsi le letsatsi, e ka ka lokisoa le bitsoa li-hormone ikutloe. Ke tsela eo, ketsahalo ena e hlokomela ka ho feta 80% ea batho ba sebediswa sehlahiswa.

Ka kakaretso, aromatase inhibitors - lithethefatsi tsebahalang lekana. generating disampole boraro blockers "Anastrozole", 'me hamorao "vorozole" le
'Letrozole', ba ile ba bōptjoa ka lihlahisoa tsa meleng e ka pele le la bobeli le hore re phekoloe hasane receptor ea HIV le kankere ea matsoele.

"Krizin"

Bakeng sa weightlifters maraka diokobatsi hape e fana ka 5,7-digidroksiflavon ( "Krizin"), e leng baatlelete sebelisa ka tekanyetso e phahameng haholo. Ho na le thepa antiaromatazatnymi le hlahisoang ka mefuta e 'meli - MRM-Chrysin, accommodating 500 mg, ka ho ya ka komiki se nang sekoli krizina le SciFit-Chrysin ES, accommodating halofo ntho mafolofolo.

litla-morao tsa ke jwa ba ne ba sa senola, empa e lokela ho a hopola hore e tsohle dintho le litokisetso le bohato antiaromatazatnym, ba nang le bokhoni ba ho baka kotsi 'meleng le semathi tsotehang. Ho feta moo, ba ile ba ba ka, "List of dintho tse thibetsoeng le mekhoa."

Reviews

bodybuilders ba bangata ba re hore, motheong oa boiphihlelo le "letrozole" ( "Femara"), ba etsa qeto ena: sehlahisoa ena, ke ho rarolla bothata le mong (phahameng pontshi tsa estrogen bananeng,), e khothalletsa ho hlaha ha mathata a mang a mangata. Ya e le hantle, inhibitors aromatase ke tsa bohlokoa bakeng sa banna. Ka mor'a hore tsohle, 'mele (banna ka ho khetheha) sebedisa estrogen bananeng ho boloka bophelo bo botle ba boitshireletso ba mmele, boko, ho tloaelehile k'holeseterole, ka bophelo bo botle le manonyello, ligaments,' me joalo-joalo.

Baatlelete ba re estrogen bananeng ho etsa hore mochine ea 'mele ea ho hōla mesifa. Noa 2,5 mg, "letrozole" ka letsatsi ba qala ho ikutloa u hlaha kotsi e tebileng articular manonyello le ligaments, 'me ba kotsing ea ho mafu a tšoaetsanoang le ho bongata ba kokwanahloko.

baatlelete ba bangata ba lumela hore 'Letrozole' na ha sebelisoa feela bodybuilders litsebi lokisetsa peisong. Thanks ho eena, ba tlosa mokelikeli feteletseng 'meleng (bakeng sa profesionalce bophelo hobane tlhōlo hase masoabi). Ba thabela ho nka ka aromatase sesitisa. theko bona kgotsofetse haholo.

Ba bang ba baatlelete re 'Letrozole' phello e ntle 'mele esita le ho lethal dose e le ba 0.1-0.5 mg,. Ba tlaleha hore ha ho hobe le ho feta tšusumetso e nyenyane tsa inhibitors e meng, le tekanyetso bakeng sa mofuta ona wa meriana. Ba ba bolela hore subjectively, sehlahiswa e ka potlako fetola tsebetso lekwalata bophahamo ba modumo ho feta "Tamoxifen" le "Clomid". Ba ile ba boela ba pheha khang ea hore aromatase inhibitors - lithethefatsi tse theko justifies boleng.

Ba bang ba baatlelete tlaleho e ka sebelisoa blocker efe kapa efe, empa ba fuoa phahameng tlhahiso "letrozole" ka tekanyetso e nyenyane, e le sa theko e tlaase ka ho fetisisa.

"Anastrozole"

Kajeno "Anastrozole" ke blocker ratoang ka ho fetisisa. The maleewana o nkoa e le "motse." Tse ling tsa inhibitors aromatase ka famasi ba ka seoelo, ho etsa mohlala, "Anastrozole kabhi."

batho ba bangata ha boloka ka bophelo ba bona le ho khetha boleng.

Nka "Anastrozole" ho latela boemo ba sona ba estradiol. Ka lebaka leo, pele lekoa maemo estradiol ho fetola thehiloeng and analysis karolo. Karolelano ea classic litekanyetso li behoa ke 0.5 mg, ka ho ya ka letsatsi.

Matsatsi a leshome hamorao, o lokela ho hlahloba hape. Ha boemo ba estradiol tekanyetso e, ho ka etsahala ho fokotsa litekanyetso li behoa ea 0.5 mg, ka makhetlo a mabeli ka beke. Ha e ntse e phahameng, le baeti ba fihlelang ho lokela ho tsoela pele. Me ho joalo le e lokela ho ba ha e le hantle ho fihlela maemo a hlaphoheloe feletseng estradiol.

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